AKR1C3-IN-1
CAT:
804-HY-107379-03
Size:
10 mM / 1 mL
Price:
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
AKR1C3-IN-1
- CAS Number: 327092-81-9
- UNSPSC Description: AKR1C3-IN-1 is a potent, highly selective inhibitor of AKR1C3, with an IC50 of 13 nM.
- Target Antigen: 17β-HSD
- Type: Reference compound
- Related Pathways: Metabolic Enzyme/Protease
- Field of Research: Others
- Assay Protocol: https://www.medchemexpress.com/AKR1C3-IN-1.html
- Purity: 98.23
- Solubility: DMSO : ≥ 100 mg/mL
- Smiles: O=S(N1CC2=CC=CC=C2CC1)(C3=CC(C(O)=O)=CC=C3)=O
- Molecular Weight: 317.36
- References & Citations: [1]Jamieson SM, et al. 3-(3,4-Dihydroisoquinolin-2(1H)-ylsulfonyl)benzoic Acids: highly potent and selective inhibitors of the type 5 17-β-hydroxysteroid dehydrogenase AKR1C3. J Med Chem. 2012 Sep 13;55(17):7746-58.
- Shipping Conditions: Room Temperature
- Storage Conditions: -20°C, 3 years; 4°C, 2 years (Powder)
- Clinical Information: No Development Reported