EN40

• UNSPSC Description:

  EN40 is a potent, selective aldehyde dehydrogenase 3A1 (ALDH3A1) inhibitor as a covalent ligand, exhibits an IC50 value of 2 uM[1]

• Target Antigen:

  Aldehyde Dehydrogenase (ALDH)

• Type:

  Reference compound

• Related Pathways:

  Metabolic Enzyme/Protease

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/en40.html

• Purity:

  99.56

• Solubility:

  DMSO : ≥ 100 mg/mL|Ethanol : 100 mg/mL (ultrasonic)

• Smiles:

  C=CC(N1CCC(C)=C(C2=CC=CO2)C1)=O

• Molecular Weight:

  217.26

• References & Citations:

  [1]Counihan JL,et al.Chemoproteomics-Enabled Covalent Ligand Screening Reveals ALDH3A1 as a Lung Cancer Therapy Target.ACS Chem Biol. 2018 Aug 17;13(8):1970-1977

• Shipping Conditions:

  Room Temperature

• Storage Conditions:

  4°C (Powder, stored under nitrogen)

• Clinical Information:

  No Development Reported

• CAS Number:

  2094547-67-6