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Omarigliptin (MK-3102)

CAT: 1568-C13501-5mgSize: 5 mgDry Ice: YesHazardous: No
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CAT#:1568-C13501-5mgSize:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1226781-44-7
Target
DPP
Applications
Metabolism
Smiles
CS (=O) (=O) N1C=C2CN (CC2=N1) C3CC (C (OC3) C4=C (C=CC (=C4) F) F) N
Molecular Formula
C17H20F2N4O3S
Additionnal Information
Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM) . It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5) .
Storage Conditions
2 years -80 in solvent

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Alternative Products

CatalogName
S8565-01Omarigliptin (MK-3102)
MBS130583-01MK-3102, Omarigliptin [USAN], Omarigliptin (USAN/INN), SureCN827590, UNII-CVP59Q4JE1, CHEMBL2105762, MK-3102, PB39113
9599-5MK-3102
A13310-50MK-3102 50mg
A13310-500MK-3102 500mg
A13310-100MK-3102 100mg
A13310-10MK-3102 10mg
A13310-5MK-3102 5mg
A13310-1MK-3102 1mg
A13310-25MK-3102 25mg

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