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Omarigliptin (MK-3102)

CAT: 0957-S8565-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S8565-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM) . It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5) .
CAS Number
1226781-44-7
Target
DPP
Activity
Metabolism
Molecular Formula
C17H20F2N4O3S
Storage Conditions
2 years -80 in solvent