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Mozavaptan (hydrochloride)

CAT: 1568-C03484-25mgSize: 25 mgDry Ice: NoHazardous: No
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CAT#:1568-C03484-25mgSize:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
138470-70-9
Synonyms
OPC 31260 HCl
Target
Vasopressin Receptor
Applications
GPCR & G Protein
Molecular Formula
C27H29N3O2.ClH
Additionnal Information
Mozavaptan hydrochloride (OPC 31260 HCl), a benzazepine derivative is a potent, selective, competitive, and orally active antagonist of vasopressin V2 receptor with an IC50 value of 14 nM. Mozavaptan hydrochloride shows ~85-fold selectivity for V2 receptor over V1 receptor. Mozavaptan hydrochloride has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment.