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STL127705

CAT: 0957-E4784-25mgSize: 25 mgDry Ice: NoHazardous: No
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CAT#:0957-E4784-25mgSize:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1326852-06-5
Molecular Formula
C22H20FN5O4
Additionnal Information
STL127705 is a potent small molecule inhibitor of Ku70/80 heterodimer protein with an IC50 of 3.5 μM. It disrupts Non-Homologous End-Joining (NHEJ) by preventing DNA binding and inhibiting DNA-PKCS activation. It exhibits anticancer activity by inducing apoptosis and inhibiting cell proliferation.