Products for Research Use Only

CAY10566

CAT: 0957-E1227-100mgSize: 100 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-E1227-100mgSize:100 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
944808-88-2
Target
SCD
Applications
Metabolism
Molecular Formula
C18H17ClFN5O2
Additionnal Information
CAY10566 is a potent, orally bioavailable and selective inhibitor of stearoyl-CoA desaturase1 (SCD1) with IC50 of 4.5 and 26 nM in mouse and human enzymatic assays, respectively. It also demonstrates excellent cellular activity in blocking the conversion of saturated long-chain fatty acid-CoAs (LCFA-CoAs) to monounsaturated LCFA-CoAs in HepG2 cells.