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Evocalcet

CAT: 0957-E0359-5mgSize: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-E0359-5mgSize:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
870964-67-3
Synonyms
KHK7580
Target
CaSR
Applications
GPCR & G Protein
Molecular Formula
C24H26N2O2
Additionnal Information
Evocalcet (KHK7580) is an novel oral calcimimetic agent which acts via allosteric activation of the calcium sensing receptor (CaSR) . Evocalcet (0, 20 and 60 nM) dose-dependently increases cytoplasmic [Ca2+] concentrations with an EC50 value of 92.7 nM in hCaR-HEK293 cells.
Storage Conditions
3 years -20°C powder