SGC-CBP30

• CAS Number :

  1613695-14-9

• SKU :

  C12552-10mg

• Target :

  Epigenetic Reader Domain

• Applications :

  Epigenetics

• Smiles :

  CC1=C (C (=NO1) C) C2=CC3=C (C=C2) N (C (=N3) CCC4=CC (=C (C=C4) OC) Cl) CC (C) N5CCOCC5

• Molecular Formula :

  C28H33ClN4O3

• Additionnal Information :

  SGC-CBP30 is a potent CREBBP/EP300 inhibitor with IC50 of 21 nM and 38 nM in cell-free assays, respectively. Exhibits 40-fold and 250-fold selectivity for CBP over the first BRD of BRD4 (BRD4 (1) ) and BRD4 (2) respectively.

• Storage Conditions :

  2 years -80 in solvent