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Bilastine-d6

CAT: 0804-HY-14447S-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-14447S-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Bilastine-d6 is the deuterium labeled Bilastine. Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria[1][2].
CAS Number
1215358-58-9
UNSPSC
12352005
Target
Histamine Receptor; Isotope-Labeled Compounds
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling; Others
Field of Research
Inflammation/Immunology; Endocrinology
Purity
97.12
Solubility
DMSO : 10 mg/mL (ultrasonic; warming)
Smiles
CCOCCN1C(C2CCN(CC2)CCC3=CC(C(C([2H])([2H])[2H])(C([2H])([2H])[2H])C(O)=O)=CC=C3)=NC4=CC=CC=C41
Molecular Formula
C28H31D6N3O3
Molecular Weight
469.65
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216. |[2]Corcostegui, R., et al., Preclinical pharmacology of bilastine, a new selective histamine H1 receptor antagonist: receptor selectivity and in vitro antihistaminic activity. Drugs R D, 2005. 6 (6) : p. 371-84.; Jauregizar, N., et al., Pharmacokinetic-pharmacodynamic modelling of the antihistaminic (H1) effect of bilastine. Clin Pharmacokinet, 2009. 48 (8) : p. 543-54.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Isoform
H1 Receptor

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