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(±) -Fabesetron

CAT: 0804-HY-101638ASize: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-101638ASize:1 Each
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Description
(±) -Fabesetron ((±) -FK1052 free base) is the racemate of Fabesetron, which is a potent 5-HT3 and 5-HT4 receptor dual antagonist[1].
CAS Number
129299-72-5
Product Name Alternative
(±) -FK1052 (free base)
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Pyrido[1,2-a]indol-6_7H_-one,_8,9-dihydro-10-methyl-7-[_4-methyl-1H-imidazol-5-yl_methyl]-.html
Solubility
10 mM in DMSO
Smiles
O=C1C(CC2=C(C)N=CN2)CCC(N31)=C(C)C4=C3C=CC=C4
Molecular Formula
C18H19N3O
Molecular Weight
293.36
References & Citations
[1]Kadowaki M, et al. Effect of FK1052, a potent 5-hydroxytryptamine3 and 5-hydroxytryptamine4 receptor dual antagonist, on colonic function in vivo. J Pharmacol Exp Ther. 1993 Jul;266 (1) :74-80.|[2]Yamakuni H, et al. Probable involvement of the 5-hydroxytryptamine (4) receptor in methotrexate-induced delayed emesis in dogs. J Pharmacol Exp Ther. 2000 Mar;292 (3) :1002-7.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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