NSD2-IN-5

• Description:

  NSD2-IN-5 (Compound 198) is an NSD2 inhibitor with an IC50 value between 0.001 μM and 0.01 μM. NSD2-IN-5 can be used in cancer research[1].

• UNSPSC:

  12352005

• Target:

  Histone Methyltransferase

• Related Pathways:

  Epigenetics

• Field of Research:

  Cancer

• Smiles:

  FC(C=C1C2=NC=C(N3CCC[C@@](N)(C3)C4=CC=CC=N4)C(CN5C6=NC=NC(N)=C6N=C5)=C2)=C(C=C1)F

• Molecular Formula:

  C27H25F2N9

• Molecular Weight:

  513.54

• References & Citations:

  [1]Haibin Deng, et al. Piperidinyl-methyl-purineamines as nsd2 inhibitors and anti-cancer agents. WO2021026803A1. WIPO (PCT) . 2019-08-14.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• Isoform:

  NSD2/MMSET/WHSC1

• CAS Number:

  2604513-53-1