SGC-GAK-1
CAT:
804-HY-122186-03
Size:
10 mg
Price:
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
SGC-GAK-1
- CAS Number: 2226517-76-4
- UNSPSC Description: SGC-GAK-1 is a potent, selective cyclin G-associated kinase (GAK) inhibitor with a Ki of 3.1 nM. SGC-GAK-1 is a chemical probe for GAK[1].
- Target Antigen: Cyclin G-associated Kinase (GAK)
- Type: Reference compound
- Related Pathways: Cell Cycle/DNA Damage
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/SGC-GAK-1.html
- Purity: 99.92
- Solubility: DMSO : 41.67 mg/mL (ultrasonic)
- Smiles: COC1=C(C(OC)=CC(NC2=CC=NC3=CC=C(C=C23)Br)=C1)OC
- Molecular Weight: 389.24
- References & Citations: [1]Asquith CRM, et al. SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK). J Med Chem. 2019 Feb 26.
- Shipping Conditions: Room Temperature
- Storage Conditions: -20°C, 3 years; 4°C, 2 years (Powder)
- Clinical Information: No Development Reported