[Dmt1]DALDA

CAT: 0931-TP3815-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-TP3815-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
255861-98-4
Target
Opioid Receptor
Related Pathways
GPCR/G Protein|||Neuroscience|||Endocrinology/Hormones
Bioactivity
[Dmt1]DALDA is a potent and long-lasting analgesic that interacts with the ?-opioid receptor (mu-opioid receptor), exhibiting high affinity and selectivity. It acts as a full agonist for hMOR (Kd= 0.199 nM) and hDOR, yet only serves as a partial agonist for hKOR.
Smiles
[C@@H](CC1=CC=CC=C1)(NC([C@H](NC([C@H](CC2=C(C)C=C(O)C=C2C)N)=O)CCCNC(=N)N)=O)C(N[C@@H](CCCCN)C(N)=O)=O
Molecular Formula
C32H49N9O5
Molecular Weight
639.79
Shipping Conditions
Cool pack
Storage Temperature
-20°C