Products for Research Use Only

CSNK2-IN-1

CAT: 0931-T89535-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T89535-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Casein Kinase
Related Pathways
Stem Cells, Metabolism
Bioactivity
CSNK2-IN-1 is a potent and selective inhibitor of CSNK2, exhibiting IC50 values of 1.7 nM for CSNK2A1 and 0.66 nM for CSNK2A2. It demonstrates antiviral activity against β-coronaviruses, including SARS-CoV-2 and MHV. Despite its favorable solubility, metabolic stability, and low cytotoxicity, CSNK2-IN-1 experiences a rapid decline in plasma concentration in vivo, which is insufficient for pharmacological effects. This compound is suitable for research in antiviral drug development.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C