Products for Research Use Only

EBET-1055

CAT: 0931-T87715-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T87715-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
ADC Cytotoxin, PROTACs, Epigenetic Reader Domain
Related Pathways
Antibody-drug Conjugate/ADC Related, Chromatin/Epigenetic, PROTAC
Bioactivity
EBET-1055 is a degrader of bromodomain and extra-terminal (BET) proteins, consisting of a BET inhibitor (EBET-590), an E3 ubiquitin ligase ligand, and connectors. It effectively inhibits the growth of pancreatic ductal adenocarcinoma (PDAC) and also modulates cancer-associated fibroblast (CAF) activity, enhancing all reporter gene activities in organoid co-cultures [1].
Molecular Formula
C51H54N8O9
Molecular Weight
923.02
Shipping Conditions
Ice Packs
Storage Temperature
-20°C