HY-078020

• Target:

  Histamine Receptor|||AChR

• Related Pathways:

  GPCR/G Protein|||Neuroscience|||Immunology/Inflammation

• Bioactivity:

  HY-078020 (compound III-4), a selective and orally active histamine H1 receptor antagonist, demonstrates an IC50 of 24.12 nM. It exhibits anti-inflammatory effects in allergic diseases [1].

• Smiles:

  ClC=1C=C2C(C(C=3C(CC2)=CC=CN3)=C4CCN(CCCC5=CC(C(C(O)=O)(C)C)=CC=C5)CC4)=CC1

• Molecular Formula:

  C32H35ClN2O2

• Molecular Weight:

  515.09

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2756222-90-7