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GPR40 agonist 7

CAT: 0931-T86521-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T86521-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1821647-46-4
Target
GPCR
Related Pathways
GPCR/G Protein, Endocrinology/Hormones
Bioactivity
Compound 1, also known as GPR40 agonist 7, is an orally active agonist of the G protein-coupled receptor 40 (GPR40) . It effectively enhances the secretion of insulin and GLP-1, exhibiting a hypoglycemic effect in vivo with an ED 50 of 0.58 mg/kg [1].
Smiles
C(C(O)=O)[C@@H]1N(C[C@H](OCCCOC)[C@H]1C)C2=CC=C(O[C@H]3[C@H](C)CN(CC3)C=4C=C(OC)N=CC4Cl)C=C2
Molecular Formula
C29H40ClN3O6
Molecular Weight
562.1
Shipping Conditions
Ice Packs
Storage Temperature
-20°C