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Edonentan hydrate

CAT: 0931-T86338-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T86338-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
264609-13-4
Target
Endothelin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
Edonentan (BMS 207940) hydrate effectively blocks the endothelin A (ETA) receptor as a potent and selective antagonist, featuring a K i of 10 pM. It exhibits complete (100%) oral bioavailability in rats [1].
Smiles
C(N(C(CC(C)(C)C)=O)C)C1=C(C=CC(=C1)C2=NC=CO2)C3=C(S(NC=4C(C)=C(C)ON4)(=O)=O)C=CC=C3.O
Molecular Formula
C28H34N4O6S
Molecular Weight
554.66
Shipping Conditions
Ice Packs
Storage Temperature
-20°C