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AR antagonist 5

CAT: 0931-T85717-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T85717-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2902679-53-0
Target
Androgen Receptor
Related Pathways
Endocrinology/Hormones
Bioactivity
Compound 30a, known as AR Antagonist 5, is a selective androgen receptor (AR) antagonist that demonstrates an IC 50 value of 134.8 nM. It exhibits favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure [1].
Smiles
C([C@](C(NC=1C=C(C(F)(F)F)C(C#N)=NC1)=O)(C)O)N2CC3N(C(C3)C2)C4=CC=C(C#N)C=C4
Molecular Formula
C23H21F3N6O2
Molecular Weight
470.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C