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PRT543

CAT: 0931-T84861-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T84861-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1989620-03-2
Target
Others, Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
PRT543 is a potent selective inhibitor of the protein arginine methyltransferase 5 (PRMT5), showing a wide range of antitumor activities in vitro and in vivo. The compound also showed an inhibitory effect on methyltransferase activity of the PRMT5/MEP50 complex with an IC50 value of 10.8 nM.
Smiles
O[C@H]1[C@H](N2C=3C(C=C2)=C(N)N=CN3)O[C@]([C@H](O)C4=CC=C(Cl)C=C4)([C@H]1O)[H]
Molecular Formula
C17H17ClN4O4
Molecular Weight
376.79
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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Alternative Products

CatalogName
C01787-5mgPRT543
A24356-50PRT543 (PRMT5-IN-35) 50mg
A24356-10PRT543 (PRMT5-IN-35) 10mg
A24356-100PRT543 (PRMT5-IN-35) 100mg
A24356-5PRT543 (PRMT5-IN-35) 5mg

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