Leumorphin, human

• Target:

  Opioid Receptor

• Related Pathways:

  GPCR/G Protein|||Endocrinology/Hormones|||Neuroscience

• Bioactivity:

  Leumorphin, human, is a potent agonist of the kappa opioid receptor (? opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-longitudinal muscle preparation [1].

• Smiles:

  C ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@H] (CC1=CC=CC=C1) NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@@H] (NC ([C@H] (CC2=CC=CC=C2) NC (CNC (CNC ([C@H] (CC3=CC=C (O) C=C3) N) =O) =O) =O) =O) CC (C) C) =O) CCCNC (=N) N) =O) CCCNC (=N) N) =O) CCC (N) =O) =O) =O) CCCCN) =O) [C@@H] (C) C) =O) C (C) C) =O) [C@@H] (C) O) =O) CCCNC (=N) N) =O) CO) =O) CCC (N) =O) =O) CCC (O) =O) =O) CC (O) =O) (=O) N4[C@H] (C (N[C@H] (C (N[C@H] (C (N[C@@H] (CC5=CC=C (O) C=C5) C (N[C@H] (C (NCC (N[C@H] (C (N[C@H] (C (N[C@@H] (CC6=CC=CC=C6) C (N[C@H] (C (N[C@H] (C (O) =O) C) =O) CC (O) =O) =O) =O) CC (C) C) =O) CCC (O) =O) =O) =O) CO) =O) =O) C) =O) CC (N) =O) =O) CCC4

• Molecular Formula:

  C150H224N42O46

• Molecular Weight:

  3351.64

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  88846-98-4