Products for Research Use Only

Ac-RYYRIK-NH2 TFA

CAT: 0931-T75907-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T75907-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Opioid Receptor
Related Pathways
GPCR/G Protein, Endocrinology/Hormones, Neuroscience
Bioactivity
Ac-RYYRIK-NH2 TFA acts as both a potent partial agonist for ORL1 when transfected in CHO cells (K d = 1.5 nM) and an endogenous ligand of ORL1. Moreover, it serves as a specific antagonist that inhibits G protein activation and competitively blocks the stimulation of [35S]-GTPγS binding to G proteins by nociceptin/orphanin FQ (noc/OFQ) in rat brain membranes and sections [1].
Molecular Formula
C46H71F3N14O11
Molecular Weight
1053.13
Shipping Conditions
Ice Packs
Storage Temperature
-20°C