Products for Research Use Only

BQ-123 TFA

CAT: 0931-T73877-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T73877-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Others, Endothelin Receptor
Related Pathways
GPCR/G Protein, Others
Bioactivity
BQ-123 TFA, a potent and selective endothelin A (ETA) receptor antagonist, demonstrates an IC50 of 7.3 nM and a Ki of 25 nM. It effectively inhibits endothelin-1-induced proliferation of human pulmonary artery smooth muscle cells and reduces blood pressure in various rat hypertension models [1] [2] [3].
Molecular Formula
C33H43F3N6O9
Molecular Weight
724.72
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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