BQ-123 TFA
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
BQ-123 TFA
Target :
Others|||Endothelin ReceptorRelated Pathways :
GPCR/G Protein|||OthersBioactivity :
BQ-123 TFA, a potent and selective endothelin A (ETA) receptor antagonist, demonstrates an IC50 of 7.3 nM and a Ki of 25 nM. It effectively inhibits endothelin-1-induced proliferation of human pulmonary artery smooth muscle cells and reduces blood pressure in various rat hypertension models [1] [2] [3].Molecular Formula :
C33H43F3N6O9Molecular Weight :
724.72Shipping Conditions :
Cool packStorage Temperature :
-20°C
