BI-2081

• Target:

  Others|||GPCR

• Related Pathways:

  GPCR/G Protein|||Endocrinology/Hormones|||Others

• Bioactivity:

  BI-2081, a GPR40 (FFAR1) partial agonist with an EC50 of 4 nM, promotes glucose-dependent insulin secretion and lowers plasma glucose levels. This compound is utilized in metabolic disease research, specifically targeting type 2 diabetes.

• Smiles:

  O ([C@H]1C=2C (=C (C=CC2F) C3=C (C) C=C (OCCC (C) (C) O) C=C3C) CC1) C=4C=C5C (=CC4) [C@H] (CC (O) =O) CO5

• Molecular Formula:

  C32H35FO6

• Molecular Weight:

  534.62

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1458656-71-7