RS-102221

• Target :

  5-HT Receptor

• Related Pathways :

  GPCR/G Protein|||Neuroscience

• Bioactivity :

  RS-102221 is a selective antagonist of the 5-HT2C receptor with a K i of 10 nM, demonstrating nearly 100-fold more selectivity for the 5-HT2C receptor over the 5-HT2A and 5-HT2B receptors. This compound not only has the potential to promote the differentiation of new nerve cells but also increases food intake and weight gain in rats.

• Smiles :

  O=C1NC(=O)C2(N1)CCN(CCCCC(=O)C3=CC(NS(=O)(=O)C4=CC=C(C=C4)C(F)(F)F)=C(OC)C=C3OC)CC2

• Molecular Formula :

  C27H31F3N4O7S

• Molecular Weight :

  612.62

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  185376-97-0