(E/Z) -Ensifentrine

• Target :

  Others|||PDE

• Related Pathways :

  Metabolism|||Others

• Bioactivity :

  (E/Z) -Ensifentrine is a potent and selective PDE3/4 inhibitor that acts as a long-acting inhibitor of the phosphodiesterase enzymes PDE-3 and PDE-4, producing both bronchodilator and anti-inflammatory effects. It is being developed by Verona Pharma as a potential treatment for asthma and hay fever and is currently in clinical trials.

• Smiles :

  O=C1N2C(C=3C(=CC(OC)=C(OC)C3)CC2)=CC(=NC4=C(C)C=C(C)C=C4C)N1CCNC(N)=O

• Molecular Formula :

  C26H31N5O4

• Molecular Weight :

  477.56

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  298680-25-8