(E/Z) -Ensifentrine

• Target:

  Others|||PDE

• Related Pathways:

  Metabolism|||Others

• Bioactivity:

  (E/Z) -Ensifentrine is a potent and selective PDE3/4 inhibitor that acts as a long-acting inhibitor of the phosphodiesterase enzymes PDE-3 and PDE-4, producing both bronchodilator and anti-inflammatory effects. It is being developed by Verona Pharma as a potential treatment for asthma and hay fever and is currently in clinical trials.

• Smiles:

  O=C1N2C (C=3C (=CC (OC) =C (OC) C3) CC2) =CC (=NC4=C (C) C=C (C) C=C4C) N1CCNC (N) =O

• Molecular Formula:

  C26H31N5O4

• Molecular Weight:

  477.56

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  298680-25-8