Ensifentrine

CAT: 0931-T25376-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-T25376-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1884461-72-6
Target
PDE
Related Pathways
Metabolism
Purity
0.9994
Bioactivity
Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for PDE3 (IC50: 0.4 nM) is 3,440 times higher than that for PDE4 (IC50: 1479 nM), that is under clinical development for the treatment of asthma and COPD and, potentially, cystic fibrosis.
Smiles
COc1cc2CCn3c(c\c(=N/c4c(C)cc(C)cc4C)n(CCNC(N)=O)c3=O)-c2cc1OC
Molecular Formula
C26H31N5O4
Molecular Weight
477.56
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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