ATR-258

CAT: 0931-T210670-01Size: 10 mgDry Ice: NoHazardous: No

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CAT#:0931-T210670-01Size:10 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

2301983-88-8

Target

Adrenergic Receptor

Related Pathways

GPCR/G Protein, Neuroscience

Bioactivity

ATR-258 is a GRK2-biased partial agonist of β2AR. It acts as a competitive antagonist of β1AR and exhibits weak partial agonist activity on β3AR at a concentration of 10 μM. ATR-258 enhances glycemic control and reduces lipid accumulation in obese mice with minimal side effects. It is applicable in research on type 2 diabetes (T2DM) .

Smiles

[C@@H](CNC(C)(C)C)(O)C=1C=C(F)C=NC1

Molecular Formula

C11H17FN2O

Molecular Weight

212.26

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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GTR19263184-01	ATR-258
A2168-5	Dovitinib (TKI-258, CHIR-258)
552471	ATR
E1884-1g	HC-258
GTR19220973-01	JG-258
XSB44389-01	BML-258

ATR-258

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