KAT6A/KAT7-IN-3

• Target:

  Histone Acetyltransferase

• Related Pathways:

  Chromatin/Epigenetic

• Bioactivity:

  KAT6A/KAT7-IN-3 (Example 191) is an inhibitor of KAT6A and KAT7. It exhibits an IC50 of 10-50 nM for KAT6A and 1 nM or less for KAT7. This compound inhibits acetylation of H3K14 and H3K23 and suppresses tumor cell proliferation, with an IC50 of 2-5 ?M for CAMA-1. KAT6A/KAT7-IN-3 is applicable in cancer research.

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C