Products for Research Use Only

EGFR-IN-107

CAT: 0931-T209547-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T209547-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
EGFR, Apoptosis
Related Pathways
Angiogenesis, JAK/STAT signaling, Tyrosine Kinase/Adaptors, Apoptosis
Bioactivity
EGFR-IN-107 (compound 3r) is an orally active EGFR inhibitor with IC50 values of 0.4333 μM for EGFRWT and 0.0438 μM for EGFRL858R/T790M. It exhibits antiproliferative activity, effectively inhibiting the proliferation of H1975 cells and inducing apoptosis (apoptosis) . EGFR-IN-107 is applicable in cancer research.
Molecular Formula
C34H36FN7O2
Shipping Conditions
Ice Packs
Storage Temperature
-20°C