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LNS8801

CAT: 0931-T206565-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T206565-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
925419-55-2
Target
Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Bioactivity
LNS8801 is an orally active agonist of the G protein-coupled estrogen receptor (GPER) . By activating GPER, LNS8801 mediates downstream signaling pathways, such as promoting cAMP production and activating CREB signaling, which results in antitumor activities like inhibiting tumor cell proliferation, inducing cell differentiation, and enhancing tumor immunogenicity. It is applicable in research across various cancers, such as melanoma, pancreatic cancer, colorectal cancer, and lung cancer, as well as studies exploring the role of GPER in normal physiological and pathological processes.
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BrC1=C([C@@H]2[C@]3([C@@](C=4C(N2)=CC=C(C(C)=O)C4)(C=CC3)[H])[H])C=C5C(=C1)OCO5
Molecular Formula
C21H18BrNO3
Molecular Weight
412.277
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-173178-01LNS8801

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