Products for Research Use Only
RegisterLogin

GJG057

CAT: 0931-T205247-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T205247-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
2761767-18-2
Target
Glutathione Peroxidase, GST
Related Pathways
Oxidation-Reduction, Metabolism
Purity
0.998
Bioactivity
GJG057 is a highly efficient and selective Leukotriene C4 synthase (LTC4S) inhibitor with an IC50 of 44 nM in human whole blood LTC4 release assays and oral activity. It demonstrates anti-inflammatory efficacy in a mouse asthma exacerbation model and can be used for the treatment of allergic inflammation.
Smiles
O=C1N(C2=CC=C(F)C(F)=C2)C3(CCN(C=4N=CN=C(OCC(F)(F)F)C4)CC3)CCC1
Molecular Formula
C21H21F5N4O2
Molecular Weight
456.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-168498-01GJG057

Popular Products