PAR-2-IN-2

• CAS Number :

  313986-65-1

• Target :

  Protease-activated Receptor|||Serine Protease

• Related Pathways :

  Proteases/Proteasome|||GPCR/G Protein

• Bioactivity :

  PAR-2-IN-2 (compound P-596) is an inhibitor of protease-activated receptor 2 (PAR-2), with an IC50 of 10.79 ?M for SLIGKV and an IC50 greater than 200 ?M for trypsin.

• Smiles :

  O=C(C1=NN2C(N=C(C=C2C(F)(F)F)C=3C=CC=CC3)=C1)N4CCN(C(=O)C=5C=CC=CC5)CC4

• Molecular Formula :

  C25H20F3N5O2

• Molecular Weight :

  479.454

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C