Products for Research Use Only

ADS1017

CAT: 0931-T204233-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T204233-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Histamine Receptor, AChR
Related Pathways
GPCR/G Protein, Immunology/Inflammation, Neuroscience
Bioactivity
ADS1017 is an antagonist of histamine receptor (histamine receptor) and muscarinic receptor (muscarinic receptor), displaying strong affinity for hH3R, hH4R, hM2R, and hM4R with pKi values of 6.8, 5.5, 7.4, and 7.2, respectively. In mouse models of pain induced by Capsaicin or Oxaliplatin, ADS1017 exhibits analgesic and anti-hyperalgesic effects.
Smiles
C1CN(CCN1CCCCCCCOC2=CC=CC=C2)CCCCN(CC3=CC=CC=C3)C(=N)N
Molecular Formula
C29H45N5O
Molecular Weight
479.701
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-170444ADS1017