SR-12062

• Bioactivity:

  SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 ?M, with complete receptor activation (Emax=100%) . Compared to the parent compound 1 (EC50=178 ?M; Emax=17%), SR-12062 shows approximately 90-fold greater potency.

• Smiles:

  C(C(N[C@@H](CC(C)C)C(O)=O)=O)N1C=2C(=CC(=CC2)C3=CC4=C(N=C3)C=CC=C4)C=C1

• Molecular Formula:

  C25H25N3O3

• Molecular Weight:

  415.48

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1623019-77-1