SR-12062

CAT: 0931-T202825-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-T202825-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1623019-77-1
Bioactivity
SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 ?M, with complete receptor activation (Emax=100%) . Compared to the parent compound 1 (EC50=178 ?M; Emax=17%), SR-12062 shows approximately 90-fold greater potency.
Smiles
C(C(N[C@@H](CC(C)C)C(O)=O)=O)N1C=2C(=CC(=CC2)C3=CC4=C(N=C3)C=CC=C4)C=C1
Molecular Formula
C25H25N3O3
Molecular Weight
415.48
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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