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Orantinib (SU6668)

CAT: 0957-S1470-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S1470-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Orantinib (TSU-68, SU6668) has greatest potency against PDGFR autophosphorylation with Ki of 8 nM in a cell-free assay, but also strongly inhibits Flk-1 and FGFR1 trans-phosphorylation, little activity against IGF-1R, Met, Src, Lck, Zap70, Abl and CDK2; does not inhibit EGFR. Phase 3.
CAS Number
252916-29-3
Synonyms
TSU-68
Target
PDGFR
Activity
Protein Tyrosine Kinase
Molecular Formula
C18H18N2O3
Storage Conditions
2 years -80 in solvent