Products for Research Use Only

ML221

CAT: 0957-S8695-01Size: 10 mgDry Ice: YesHazardous: No
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CAT#:0957-S8695-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
ML221 is a potent apelin receptor (APJ) functional antagonist in cell-based assays that is >37-fold selective over the closely related angiotensin II type 1 (AT1) receptor. The IC50 values of ML221 are 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively.
CAS Number
877636-42-5
Target
Angiotensin Receptor
Activity
GPCR & G Protein
Molecular Formula
C17H11N3O6S
Storage Conditions
2 years -80 in solvent