Products for Research Use Only
RegisterLogin

Merestinib (LY2801653)

CAT: 0957-S7014-02Size: 10 mm/ 1 mLDry Ice: YesHazardous: No
Product image 1
1 / 1
CAT#:0957-S7014-02Size:10 mm/ 1 mL
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Merestinib (LY2801653) is a type-II ATP competitive, slow-off inhibitor of Met (c-Met) tyrosine kinase with a dissociation constant (Ki) of 2 nM, a pharmacodynamic residence time (Koff) of 0.00132 min (-1) and t1/2 of 525 min. Merestinib (LY2801653) also inhibits MST1R, AXL, ROS1, MKNK1/2, FLT3, MERTK, DDR1 and DDR2 with IC50 of 11 nM, 2 nM, 23 nM, 7 nM, 7 nM, 10 nM, 0.1 nM and 7 nM, respectively.
CAS Number
1206799-15-6
Target
C-Met
Activity
Protein Tyrosine Kinase
Molecular Formula
C30H22F2N6O3
Storage Conditions
2 years -80 in solvent

Related Products

CatalogName
E7462Merestinib dihydrochloride
E7462-5mgMerestinib dihydrochloride

Alternative Products

CatalogName
MBS385090-01LY2801653 (Merestinib)
C12382-10mM/1mLMerestinib (LY2801653)
A12557-1LY2801653 (Merestinib) 1mg
A12557-500LY2801653 (Merestinib) 500mg
A12557-2LY2801653 (Merestinib) 2mg
A12557-25LY2801653 (Merestinib) 25mg
A12557-100LY2801653 (Merestinib) 100mg
A15150-2Merestinib dihydrochloride (LY2801653 dihydrochloride) 2mg
A12557-10mM-DLY2801653 (Merestinib) 10mM * 1mL in DMSO
GW3922-5mgLY2801653

Popular Products