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Brequinar Sodium

CAT: 0957-S3565-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-S3565-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Brequinar Sodium (Bipenquinate, BRQ, DUP-785, NSC 368390) is a potent and selective dihydroorotate dehydrogenase (DHODH) inhibitor with IC50 of ~20 nM and triggers differentiation in the ER-HoxA9, U937, and THP1 cells with ED50 of ~1 μM.
CAS Number
96201-88-6
Synonyms
Bipenquinate, BRQ, DUP-785, NSC 368390
Target
Dehydrogenase
Activity
Metabolism
Molecular Formula
C23H14F2NNaO2
Storage Conditions
3 years -20°C powder