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PF-4981517

CAT: 0957-S2921Size: 10 mgDry Ice: YesHazardous: No
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CAT#:0957-S2921Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PF-4981517 (CYP3cide, PF-04981517) is a potent and selective inhibitor of CYP3A4 (P450) with IC50 of 0.03 μM, exhibits >500-fold selectivity over CYP3A5 and CYP3A7.
CAS Number
1390637-82-7
Synonyms
CYP3cide, PF-04981517
Target
P450 (e.g. CYP17)
Activity
Metabolism
Molecular Formula
C26H32N8
Storage Conditions
2 years -80 in solvent