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PF-562271

CAT: 0957-S2890-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S2890-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PF-562271 (PF-00562271) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM in cell-free assays, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, except for some CDKs.
CAS Number
717907-75-0
Synonyms
PF-00562271
Target
FAK
Activity
Protein Tyrosine Kinase
Molecular Formula
C21H20F3N7O3S
Storage Conditions
2 years -80 in solvent

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