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TC-E5002 (KDM2/7-IN-1)

CAT: 0957-E1793-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-E1793-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
TC-E5002 (KDM2/7-IN-1) is a selective inhibitor of histone demethylase KDM2/7 subfamily with IC50s of 6.8, 0.2, and 1.2 μM for KDM2A, KDM7A, and KDM7B, respectively. It is selective for the KDM2/7 subfamily over KDM4A, KDM4C, KDM5A, and KDM6A/UTX with IC50s of >120, 83, 55, and 100 μM, respectively. It exhibits antiproliferative activity, indicating its potential as an anticancer agent.
CAS Number
1453071-47-0
Synonyms
KDM2/7-IN-1
Target
Histone Demethylase
Activity
Epigenetics
Molecular Formula
C15H27NO4