Products for Research Use Only

Masitinib mesylate

CAT: 0957-E0814Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0957-E0814Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
Masitinib mesylate (AB-1010 mesylate) is a potent, orally bioavailable, and selective inhibitor of c-Kit with IC50 of 200 nM for human recombinant c-Kit, also inhibits PDGFRα/β with IC50s of 540/800 nM, Lyn with IC50 of 510 nM for LynB, and, to a lesser extent, FGFR3 and FAK.
CAS Number
1048007-93-7
Synonyms
AB-1010 mesylate
Target
C-Kit
Activity
Protein Tyrosine Kinase
Molecular Formula
C28H30N6OS.CH4O3S
Storage Conditions
3 years -20°C powder