ELA-21 (human)

• Description:

  High affinity apelin receptor agonist. Binds apelin receptors in left ventricle from normal and pulmonary arterial hypertensive (PAH) hearts (pKi values are 9.31 and 9.46, respectively) . Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates β-arrestin recruitment in vitro.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  2587.12

• Molecular Formula:

  C112H184N40O25S3

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  2245073-05-4