[Arg14, Lys15]Nociceptin

• Description:

  Highly potent and selective NOP receptor agonist (EC50 = 1 nM) . Displays > 875-fold selectivity over opioid receptors (IC50 values are 0.32, 280, > 10000 and 1500 for NOP, μ, δ and κ receptors respectively) . Longer lasting and 30-fold more potent than nociceptin in vivo; pronociceptive and inhibits locomotor activity.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  1909.18

• Molecular Formula:

  C82H137N31O22

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  236098-40-1