(d (CH2) 51, Tyr (Me) 2, Arg8) -Vasopressin

• Description:

  Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively) . Exhibits potent and prolonged antivasopressor activity and induces anxiolytic-like effects in the dorsal, but not ventral, hippocampus in vivo.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  1151.38

• Molecular Formula:

  C52H74N14O12S2

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  73168-24-8