(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin

• UNSPSC Description:

  (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) is a specific antagonist of vasopressin V1a receptor, with a pA2 of 6.71[1].

• Target Antigen:

  Vasopressin Receptor

• Type:

  Peptides

• Related Pathways:

  GPCR/G Protein

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Cardiovascular Disease

• Assay Protocol:

  https://www.medchemexpress.com/d-ch2-51-tyr-me-2-dab5-arg8-vasopressin.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C1CC2(CCCCC2)SSC[C@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](N1)CC3=CC=C(C=C3)OC)=O)CC4=CC=CC=C4)=O)CCC(N)=O)=O)CCN)=O)C(N5[C@@H](CCC5)C(N[C@H](C(NCC(N)=O)=O)CCCNC(N)=N)=O)=O

• Molecular Weight:

  1137.38

• References & Citations:

  [1]Chan WY, et, al. Discovery and design of novel and selective vasopressin and oxytocin agonists and antagonists: the role of bioassays. Exp Physiol. 2000 Mar;85 Spec No:7S-18S.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  176714-12-8