(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin

(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin

• CAS Number: 176714-12-8
• UNSPSC Description: (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) is a specific antagonist of vasopressin V1a receptor, with a pA2 of 6.71[1].
• Target Antigen: Vasopressin Receptor
• Type: Peptides
• Related Pathways: GPCR/G Protein
• Applications: Neuroscience-Neuromodulation
• Field of Research: Cardiovascular Disease
• Assay Protocol: https://www.medchemexpress.com/d-ch2-51-tyr-me-2-dab5-arg8-vasopressin.html
• Solubility: 10 mM in DMSO
• Smiles: O=C1CC2(CCCCC2)SSC[C@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](N1)CC3=CC=C(C=C3)OC)=O)CC4=CC=CC=C4)=O)CCC(N)=O)=O)CCN)=O)C(N5[C@@H](CCC5)C(N[C@H](C(NCC(N)=O)=O)CCCNC(N)=N)=O)=O
• Molecular Weight: 1137.38
• References & Citations: [1]Chan WY, et, al. Discovery and design of novel and selective vasopressin and oxytocin agonists and antagonists: the role of bioassays. Exp Physiol. 2000 Mar;85 Spec No:7S-18S.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported