LSD1-IN-20

• Description:

  Lsd1-in-20 is a potent dual inhibitor of LSD1/G9a with Ki values of 0.44 and 0.68 μM, respectively. LSD1-IN-20 showed antiproliferative activity against THP-1 leukemia cells and MDA-MB-231 breast cancer cells in vitro, with IC50 of 0.51 and 1.60 μM, respectively, at 72 h.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  478.63

• Molecular Formula:

  C27H38N6O2

• Notes:

  Research use only, not for human use.

• Receptor:

  Histone Demethylase

• CAS Number:

  1239589-91-3