TUG-499

• Description :

  TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39) . It shows higher affinity for FFAR1 or GPR40 relative to related receptors FFA2, FFA3, and the nuclear receptor PPARγ, as well as various other receptors, ion channels, and transporter proteins. TUG-499 is useful for studying Type 2 diabetes.

• CAS Number :

  1206629-08-4

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  320.17

• Molecular Formula :

  C16H11Cl2NO2

• Notes :

  Research use only, not for human use.

• Receptor :

  GPR | PPAR