TUG-499

• Description:

  TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39) . It shows higher affinity for FFAR1 or GPR40 relative to related receptors FFA2, FFA3, and the nuclear receptor PPARγ, as well as various other receptors, ion channels, and transporter proteins. TUG-499 is useful for studying Type 2 diabetes.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  320.17

• Molecular Formula:

  C16H11Cl2NO2

• Notes:

  Research use only, not for human use.

• Receptor:

  GPR | PPAR

• CAS Number:

  1206629-08-4